Blueprint
FORM 6-K
SECURITIES
AND EXCHANGE COMMISSION
Washington,
D.C. 20549
Report
of Foreign Issuer
Pursuant
to Rule 13a-16 or 15d-16 of
the
Securities Exchange Act of 1934
For the
month of January 2018
Commission
File Number: 001-11960
AstraZeneca PLC
1
Francis Crick Avenue
Cambridge
Biomedical Campus
Cambridge
CB2 0AA
United
Kingdom
Indicate
by check mark whether the registrant files or will file annual
reports under cover of Form 20-F or Form 40-F.
Form
20-F X Form 40-F __
Indicate
by check mark if the registrant is submitting the Form 6-K in paper
as permitted by Regulation S-T Rule 101(b)(1):
Indicate
by check mark if the registrant is submitting the Form 6-K in paper
as permitted by Regulation S-T Rule 101(b)(7): ______
Indicate
by check mark whether the registrant by furnishing the information
contained in this Form is also thereby furnishing the information
to the Commission pursuant to Rule 12g3-2(b) under the Securities
Exchange Act of 1934.
Yes __
No X
If
“Yes” is marked, indicate below the file number
assigned to the Registrant in connection with Rule 12g3-2(b):
82-_____________
AstraZeneca PLC
INDEX
TO EXHIBITS
ASTRAZENECA'S
FASENRA RECEIVES APPROVAL IN JAPAN
19 January 2018 07:00 GMT
FASENRA RECEIVES APPROVAL
IN JAPAN
Approval based on Phase III WINDWARD programme that demonstrated
significant reductions in asthma exacerbations, improvements in
lung function and
reductions in oral corticosteroid use from baseline, versus
placebo
Fasenra is the first approved respiratory biologic with an
8-week
maintenance dosing schedule
AstraZeneca
and its global biologics research and development arm, MedImmune,
today announced that the Japanese Ministry of Health, Labour and
Welfare has approved Fasenra (benralizumab) as an add-on
treatment for bronchial asthma in patients who continue to
experience asthma exacerbations despite treatment with high-dose
inhaled corticosteroid and other asthma controllers.
The approval is based on the results from the WINDWARD programme,
including the pivotal Phase III exacerbation trials,
SIROCCO
and CALIMA,
and the Phase III oral corticosteroid (OCS)-sparing trial,
ZONDA.1
Fasenra
will be available as a fixed-dose
subcutaneous injection in a prefilled syringe administered once
every four weeks for the first three doses, and then once every
eight weeks thereafter.1
Sean
Bohen, Executive Vice President, Global Medicines Development and
Chief Medical Officer at AstraZeneca, said: "The approval of
Fasenra, our first
respiratory biologic medicine, in Japan closely follows the recent
US and EU decisions and brings us another step closer to achieving
our ambition of transforming care for severe asthma patients around
the world."
Fasenra binds directly to the IL-5a receptor on eosinophils, a
type of white blood cell that are a normal part of the body's
immune system,2 and attracts natural
killer cells to induce direct, rapid and near-complete depletion of
eosinophils via apoptosis (programmed cell death).5,6,7 Elevated levels
of eosinophils, seen in about half of severe asthma patients,
impact airway inflammation and airway hyper-responsiveness,
resulting in increased asthma severity and symptoms, decreased lung
function and increased risk of exacerbations.3,4
The
Japanese approval follows US FDA approval in November 2017 and
European Commission marketing authorisation in January 2018.
Interactions with regulatory authorities in the rest of the world
are on-going.
About Severe Asthma
Asthma
affects approximately 315 million individuals worldwide. Up to 10%
of asthma patients have severe asthma, which may be uncontrolled
despite high doses of standard-of-care asthma controller medicines
and can require the use of chronic OCS.3,9,10
Severe, uncontrolled asthma is debilitating and potentially fatal
with patients experiencing frequent exacerbations and significant
limitations on lung function and quality of
life.11,12,13
Severe, uncontrolled asthma has higher
risk of mortality than severe asthma.12,14
Severe,
uncontrolled asthma can lead to a dependence on OCS, with systemic
steroid exposure potentially leading to serious short- and
long-term adverse effects including weight gain, diabetes,
osteoporosis, glaucoma, anxiety, depression, cardiovascular disease
and immunosuppression.10,15,16,17,18 There
is also a significant physical and socio-economic burden of severe,
uncontrolled asthma with these patients accounting for 50% of
asthma-related costs.19
About Fasenra (benralizumab)
Fasenra is a monoclonal antibody that recruits natural
killer cells to induce direct, rapid and near-complete depletion of
eosinophils.7,20 Depletion of
circulating eosinophils is rapid, with an onset of action within 24
hours as confirmed in early Phase I/II trials.7,20,21 Eosinophils
are the biological effector cells in approximately 50% of asthma
patients, leading to frequent exacerbations, impaired lung function
and asthma symptoms.3,4
Fasenra is now approved in the US, EU and Japan, and
under regulatory review in several other
jurisdictions.
Fasenra is the foundation of AstraZeneca's respiratory
biologics portfolio of potential new medicines targeting underlying
causes of respiratory disease. Fasenra is also being evaluated in
chronic obstructive pulmonary disease (COPD) with data readout
expected in the second half of 2018.22
Fasenra was developed by AstraZeneca with MedImmune, the
company's global biologics research and development arm and is
in-licensed from BioWa, Inc., a wholly-owned subsidiary of Kyowa
Hakko Kirin Co., Ltd., Japan.
About the WINDWARD Programme
The
WINDWARD programme in asthma is made up six Phase III trials,
including SIROCCO, CALIMA, ZONDA, BISE, BORA and
GREGALE.22
The two pivotal trials SIROCCO and
CALIMA, are
randomised, double-blinded, parallel-group, placebo-controlled
trials designed to evaluate the efficacy and safety of a regular,
subcutaneous administration of Fasenra (fixed 30mg dose) for up to
56-weeks in exacerbation-prone adult and adolescent patients 12
years of age and older.5,6
A total
of 2,510 patients (1,204 in SIROCCO and 1,306 in CALIMA) received
standard-of-care medicines (including high-dosage inhaled
corticosteroids and long-acting beta2-agonists) and
were randomised globally to receive either Fasenra 30mg every 4-weeks;
Fasenra 30mg every 4-weeks
for the first three doses followed by 30mg every 8-weeks; or
placebo administered via subcutaneous injection using an
accessorised pre-filled syringe.5,6,23
In
SIROCCO and CALIMA, patients with severe, uncontrolled eosinophilic
asthma receiving Fasenra
experienced a significant reduction in asthma exacerbations and
improvement in their lung function and asthma symptoms compared to
patients receiving placebo, on top of their standard
medicines.5,6 The most commonly
reported adverse reactions during treatment were headache (8%) and
pharyngitis (3%). Other common adverse reactions included fever,
hypersensitivity reactions and injection site
reactions.1,5,6
A
pooled post-hoc analysis of
the SIROCCO and CALIMA trials, demonstrated an association between
enhanced Fasenra efficacy
and certain easily identifiable clinical features of severe
eosinophilic asthma, including baseline blood eosinophil counts,
history of more frequent exacerbations, chronic OCS use and a
history of nasal polyposis.23
The
third registrational trial, ZONDA,
demonstrated a statistically-significant and clinically-meaningful
reduction in daily-maintenance OCS use compared with placebo for
patients with severe, uncontrolled OCS-dependent eosinophilic
asthma receiving Fasenra. The results were
published in the
New England Journal of Medicine in May 2017.24
In
addition to WINDWARD, the Phase III VOYAGER programme is currently
underway, which is evaluating the efficacy and safety of
Fasenra in patients
with severe COPD.22
About AstraZeneca in Respiratory Disease
Respiratory
disease is one of AstraZeneca's main therapy areas, and
the Company has a growing portfolio of medicines that reached more
than 18 million patients in 2017. AstraZeneca's aim is to transform
asthma and COPD treatment through inhaled combinations at the
core of care, biologics for the unmet needs of specific patient
populations, and scientific advancements in disease
modification.
The
Company is building on a 40-year heritage in respiratory disease
and AstraZeneca's capability in inhalation technology spans
pressurised metered-dose inhalers and dry powder inhalers, as well
as the Aerosphere Delivery
Technology. The company's biologics include Fasenra, (anti-eosinophil,
anti-IL-5rɑ), which is now approved in the US, EU, Japan, and
is under regulatory review in other jurisdictions, and tezepelumab
(anti-TSLP), which successfully achieved its Phase IIb primary and
secondary endpoints and has initiated Phase III. AstraZeneca's
research is focused on addressing underlying disease drivers
focusing on the lung epithelium, lung immunity and lung
regeneration.
About MedImmune
MedImmune
is the global biologics research and development arm of
AstraZeneca, a global, innovation-driven biopharmaceutical business
that focuses on the discovery, development and commercialisation of
small molecule and biologic prescription medicines. MedImmune is
pioneering innovative research and exploring novel pathways across
Oncology, Respiratory, Cardiovascular & Metabolic Diseases, and
Infection and Vaccines. The MedImmune headquarters is located in
Gaithersburg, Md., one of AstraZeneca's three global R&D
centres, with additional sites in Cambridge, UK and Mountain View,
Calif. For more information, please visit www.medimmune.com
About AstraZeneca
AstraZeneca is a global, science-led biopharmaceutical company that
focuses on the discovery, development and commercialisation of
prescription medicines, primarily for the treatment of diseases in
three therapy areas - Oncology, Cardiovascular & Metabolic
Diseases and Respiratory. The Company also is selectively active in
the areas of autoimmunity, neuroscience and infection. AstraZeneca
operates in over 100 countries and its innovative medicines are
used by millions of patients worldwide.
For more information, please visit www.astrazeneca.com
and follow us on Twitter
@AstraZeneca.
Media
Relations
|
|
|
Esra
Erkal-Paler
|
UK/Global
|
+44 203
749 5638
|
Karen
Birmingham
|
UK/Global
|
+44 203
749 5634
|
Rob
Skelding
|
UK/Global
|
+44 203
749 5821
|
Matt
Kent
|
UK/Global
|
+44 203
749 5906
|
Gonzalo
Viña
|
UK/Global
|
+44 203
749 5916
|
Jacob
Lund
|
Sweden
|
+46
8 553 260 20
|
Michele
Meixell
|
US
|
+1 302
885 2677
|
|
|
|
Investor
Relations
|
|
|
Thomas
Kudsk Larsen
|
|
+44 203
749 5712
|
Craig
Marks
|
Finance,
Fixed Income, M&A
|
+44
7881 615 764
|
Henry
Wheeler
|
Oncology
|
+44 203
749 5797
|
Mitchell
Chan
|
Oncology;
Other
|
+1 240
477 3771
|
Christer
Gruvris
|
Brilinta; Diabetes
|
+44 203
749 5711
|
Nick
Stone
|
Respiratory;
Renal
|
+44 203
749 5716
|
US toll
free
|
|
+1 866
381 7277
|
Adrian Kemp
Company Secretary
AstraZeneca PLC
References
1. Fasenra (benralizumab) Package Insert. AstraZeneca PLC,
2018.
2.
Mukherjee M, Sehmi R, Nair P. Anti-IL5 therapy for asthma and
beyond. World Allergy Organ
J. 2014;7:32.
3.
Wenzel S. Severe asthma in adults. Am J Respir Crit Care Med.
2005;172:149-160.
4.
Zhang, JY and Wenzel, SE. Tissue and BAL based biomarkers in
asthma. Immunol Allergy Clin North
Am. 2007; 27: 623-632 (vi.).
5.
FitzGerald MJ, Bleecker E, Parameswaran N, et al. Benralizumab, an
anti-interleukin-5 receptor a monoclonal antibody, as add-on
treatment for patients with severe, uncontrolled, eosinophilic
asthma (CALIMA): a randomised, double-blind, placebo-controlled
phase 3 trial. Lancet.
2016. Volume 388, Issue 10056, 2128 - 2141.
6.
Bleecker ER, Fitzgerald MJ, Chanez P, et al. Efficacy and safety of
benralizumab for patients with severe asthma uncontrolled with
high-dosage inhaled corticosteroids and long-acting b2-agonists
(SIROCCO): a randomised, multicentre, placebo-controlled phase 3
trial. Lancet. 2016. Volume
388, Issue 10056, 2115 - 2127.
7.
Kolbeck R, Kozhich A, Koike M, et al. MEDI-563, a humanized
anti-IL-5 receptor a mAb with enhanced antibody-dependent
cell-mediated cytotoxicity function. J Allergy Clin Immunol. 2010
Jun;125(6):1344-1353.e2.
8. Fasenra Prescribing Information. AstraZeneca
Pharmaceuticals LP.
9. To
T, Stanojevic S, Moores G, et al. Global asthma prevalence in
adults: findings from cross-sectional world health survey.
BioMed Central Public
Health. 2012: 12(204).
10. Global Initiative for Asthma (GINA).
Online appendix. Global strategy for asthma management and
prevention. Updated 2017. Available from: http://ginasthma.org/2017-gina-report-global-strategy-for-asthma-management-and-prevention/.
Last accessed November 2017.
11. Price D,
Fletcher M, van der Molen T. Asthma control and management in 8,000
European patients: the REcognise Asthma and LInk to Symptoms and
Experience (REALISE) survey. NPJ
Prim Care Respir Med 2014; 12; 24: 14009.
12. Peters
SP, Ferguson G, Deniz Y, et al. Uncontrolled asthma: a review of
the prevalence, disease burden and options for treatment.
Respir Med. 2006:
100(7):1139-51.
13. Adelphi
Real World Respiratory Disease Specific Programme. 2012-2014.
[Asthma patient data file], Bollington, UK. Unpublished raw data,
cited with permission.
14. Fernandes
AG, Souza-Machado C, Coelho RC et al. Risk factors for death in
patients with severe asthma. J
Bras Pneumol. 2014; 40(4): 364-372.
15. Hyland
ME, Whalley B, Jones RC, Masoli M. A qualitative study of the
impact of severe asthma and its treatment showing that treatment
burden is neglected in existing asthma assessment scales.
Qual Life Res. 2015
Mar;24(3):631-9. doi: 10.1007/s11136-014-0801-x. Epub 2014 Sep
9.
16. Global Initiative for Asthma (GINA).
Online appendix. Global strategy for asthma management and
prevention. Updated 2017. Available from: http://ginasthma.org/2017-gina-report-global-strategy-for-asthma-management-and-prevention/.
Last accessed December 2017.
17. Iribarren
C, Tolstykh IV, Miller MK, et al. Adult asthma and risk of coronary
heart disease, cerebrovascular disease, and heart failure: a
prospective study of 2 matched cohorts. Am J Epidemiol.
2012;176:1014-1024.
18. Zazzali
JL, Broder MS, Omachi TA, Chang E, Sun GH, Raimundo K. Risk of
corticosteroid-related adverse events in asthma patients with high
oral corticosteroid use. Allergy
Asthma Proc. 2015 Jul-Aug;36(4):268-74. doi:
10.2500/aap.2015.36.3863.
19. World Allergy Organization (WAO). The
management of severe asthma: economic analysis of the cost of
treatments for severe asthma. Available from: http://www.worldallergy.org/educational_programs/world_allergy_forum/anaheim2005/blaiss.php.
Last accessed May 2017.
20. Pham TH,
Damera G, Newbold P, Ranade K. Reductions in eosinophil biomarkers
by benralizumab in patients with asthma. Respir Med. 2016;
111:21-29.
21.
Laviolette M, Gossage DL, Gauvreau G, et al. Effects of
benralizumab on airway eosinophils in asthmatic patients with
sputum eosinophilia. J Allergy
Clin Immunol. 2013 Nov; 132(5): 1086 - 1096.e5.
22. AstraZeneca. Clinical Trials Appendix
Q2 2017 Results Update. Available at https://www.astrazeneca.com/content/dam/az/PDF/2017/H1/H1_2017_Results_Clinical_Trial_Appendix.pdf.
Last Accessed November 2017.
23.
FitzGerald JM, Bleecker ER, Menzies-Gow A, Zangrilli JG, Hirsch I,
Metcalfe P, Newbold P, Goldman M. Predictors of enhanced response
with benralizumab for patients with severe asthma: pooled analysis
of the SIROCCO and CALIMA studies. Lancet Respir Med. 2017 Sep
11.
24. Nair P,
Wenzel S, Rabe KF, Bourdin A, Lugogo NL, et al. Oral
glucocorticoid-sparing effect of benralizumab in severe asthma.
N Engl J Med. 2017;
376:2448-58.
SIGNATURES
Pursuant
to the requirements of the Securities Exchange Act of 1934, the
Registrant has duly caused this report to be signed on its behalf
by the undersigned, thereunto duly authorized.
Date:
19 January 2018
|
By: /s/
Adrian Kemp
|
|
Name:
Adrian Kemp
|
|
Title:
Company Secretary
|